Skip to main content
. 2011 Sep 5;32(10):1285–1293. doi: 10.1038/aps.2011.78

Table 3. Inhibitory effect of ATFX on TP metabolites in human liver microsomes in vitro. Data represent mean±SD of three experiments.

  KI (μmol/L) Kapp,i (μmol/L) kinact,i (min−1) kinact,i/Kapp,i (×10−5) (min−1·M−1)
3-MX 1209.2±66.3 265.88±18.81 0.0097±0.0016 3.68±0.84
1-MX 1033.2±78.9 353.29±16.20 0.0073±0.0012 2.06±0.37
1,3-DMU 1519.4±56.6 430.21±14.19 0.0047±0.0080 1.08±0.15