Table 1. Experimentally Determined Inhibitory Activity of the 10 Compounds Selected from the Virtual Screening.
compound | NSC or UC/GRI | % inhibition at 150 μM | IC50 (μM)a | hits tested | % yield of active compounds |
---|---|---|---|---|---|
1 | NSC-334943 | 61% | 135 | 81 | 2.5% |
2 | UC-521228 | 42% | ND | ||
3 | NSC-334344 | 67% | 146 | 40 | 10% |
4 | NSC-657705 | 43% | ND | ||
5 | NSC-112182 | 43% | ND | ||
6 | NSC-25812 | 41% | ND | ||
7 | NSC-176297 | 56% | ND | 25 | 16% |
8 | NSC-106893 | 68% | 95 | ||
9 | NSC-97914 | 59% | ND | ||
10 | NSC-357905 | 73% | 48 |
ND: Not Determined.