Kinome Scan Symbol	GS-9973		R406
	Kd (nM)	Selectivity (Fold)	Kd (nM)	Selectivity (Fold)
ABL1-nonphos.	8400	800	8400	560
ABL1-phos.	560	53	560	37
ALK	2900	276	240	16
AXL	1900	181	82	5
BIKE	1100	105	1900	127
BLK	420	40	25	1.7
BRK	330	31	360	24
CHEK2	40000	3810	1000	67
CSF1R	180	17	31	2.1
CSNK2A1	540	51	1400	93
CSNK2A2	110	10	1200	80
DAPK1	40000	3810	55	4
DAPK3	40000	3810	13	0.9
EGFR	1400	133	300	20
EPHA1	470	45	67	4
EPHB6	550	52	310	21
FGR	230	22	33	2.2
FLT3	320	30	0.71	0.05
FLT3-autoinhib.	40000	3810	13	0.9
GAK	1300	124	250	17
GRK4	40000	3810	450	30
HCK	410	39	150	10
HIPK1	40000	3810	820	55
HIPK3	40000	3810	3200	213
INSR	1800	171	1100	73
IRAK1	140	13	9.7	0.6
IRAK3	120	11	11	0.7
JAK1(JH1-cat.)	730	70	21	1.4
JAK2(JH1-cat.)	110	10	3.5	0.2
JAK3(JH1-cat.)	3200	305	36	2.4
JNK1	2000	190	38	3
KIT	210	20	6.8	0.5
LCK	820	78	30	2.0
LOK	40000	3810	70	5
LTK	1200	114	800	53
MA P4K2	40000	3810	670	45
MEK5	200	19	27	1.8
MERTK	3300	314	170	11
MLK1	570	54	4.3	0.3
PDGFRB	670	64	3.3	0.2
PIP5K1A	40000	3810	1900	127
PIP5K1C	40000	3810
PIP5K2B	40000	3810	1200	80
PRKR	3000	286	180	12
RET	1000	95	4.1	0.3
RIOK1	40000	3810	340	23
RIOK2	160	15	3400	227
RIOK3	40000	3810	210	14
SBK1	40000	3810	93	6
SLK	820	78	33	2.2
SRC	110	10	8.4	0.6
SRMS	910	87	610	41
SRPK1	40000	3810	590	39
SRPK3	3200	305	400	27
STK16	330	31	1.7	0.1
STK33	40000	3810	970	65
SYK	10.5	1	15	1
TAK1	490	47	49	3
TGFBR2	390	37	330	22
TNK1	86	8	25	1.7
TNK2	670	64	70	5
TYK2(JH1-cat.)	180	17	190	13
ULK3	510	49	7.1	0.5
VEGF R2	40000	3810	40	3
YES	450	43	35	2.3
YSK4	440	42	67	4
ZAP70	410	39	21	1.4