TABLE 1.
Hepatotoxicity of Hsp90 inhibitors in the TAMH cell line
Data expressed as mean ± S.D. of three independent experiments.
Compound | IC50 | LC50 |
---|---|---|
µM | ||
17-DMAG | 0.02 ± 0.01 | 0.21 ± 0.01 |
19Ph-DMAG | 4.61 ± 0.39 | 13.83 ± 3.57 |
19Me-DMAG | 8.00 ± 0.37 | 42.67 ± 0.16 |