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. 2013 Nov 1;37(5):588–599. doi: 10.1007/s12272-013-0253-9

Scheme 5.

Scheme 5

Reagents and conditions: (a) NBS, CH3CN, reflux; (b) dioxane, reflux or NaHCO3, dioxane, reflux; (c) EtOH, reflux