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. 2011 Aug 5;2(10):786–791. doi: 10.1021/ml200175q

Table 2. SAR at the R4 Position.

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a

EC50 values were calculated as an average of at least two determinations.

b

PD responses were measure at 4 h after oral administration of compounds at 30 mg/kg in a solution formulation (ethanol:propylene glycol:10% solutol = 1:1:8).