Table 2. Rat PK Propertiesa of Phenol Replacements.
| no. | iv t1/2 (min) | CL (mL/min/kg) | oral AUC (μM h) | Vss (L/kg) | po % F |
|---|---|---|---|---|---|
| 3 | 30 | 179 | 0.03 | 6.9 | 1 |
| 4 | 55 | 26 | 16 | 2.4 | 46 |
| 5 | 103 | 5 | 93 | 0.8 | 56 |
| 12 | 43 | 37 | 6 | 1.9 | 23 |
Amounts: 5 mpk iv and 20 mpk po.
| no. | iv t1/2 (min) | CL (mL/min/kg) | oral AUC (μM h) | Vss (L/kg) | po % F |
|---|---|---|---|---|---|
| 3 | 30 | 179 | 0.03 | 6.9 | 1 |
| 4 | 55 | 26 | 16 | 2.4 | 46 |
| 5 | 103 | 5 | 93 | 0.8 | 56 |
| 12 | 43 | 37 | 6 | 1.9 | 23 |
Amounts: 5 mpk iv and 20 mpk po.