Table 2. S1P Receptor Subtype Selectivity of 8a.
| EC50 (μM) | |||
|---|---|---|---|
| hS1P2 | hS1P3 | hS1P4 | hS1P5 (% eff.) |
| >25 | >25 | >50 | 4.3 (58) |
a
See the Supporting Information for experimental details (data represent an average of at least two determinations; see ref (44)).
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