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. 2011 Mar 24;2(6):424–427. doi: 10.1021/ml100309n

Table 1. IC50 Values for Inhibition of CE Transfera.

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a

IC50 values were determined using a standard bioassay described in ref (10). The IC50 value for torcetrapib was been determined by this method in ref (7a) and was reported to be 13 nM.

b

Average of three or more 10 point titrations.

c

Result of a single 10 point titration.

d

Average of two 10 point titrations.

e

Inactive indicates <50% inhibition of CETP at a concentration of 100 μM.