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. Author manuscript; available in PMC: 2014 May 12.
Published in final edited form as: Clin Pharmacol Ther. 2012 Sep 26;92(5):661–665. doi: 10.1038/clpt.2012.164

Table 1.

Variability of Kt values for hOCT2 with transfection system (data from [35] and our laboratories).

Compound Kt
(µM)
Transfection
system
Reference
Dopamine 1400 cc [53]
390 oo [54]

Histamine 940 cc [53]
1300 oo [54]

MPP 19 oo [55]
7.8 cc [56]
12 cc Unpublished
3.1 cc [57]
12.3 Unpublished
19.5 cc [58]

Norepinephrine 1500 cc [53]
1900 oo [54]

Serotonin 290 cc [53]
80 oo [54]

TEA 27 cc [59]
76 oo [55]
109 cc [60]
20 cc [61]
46 cc [17]

cc = cultured cell (HEK293 or CHO), oo = oocyte, MPP = 1-methyl-4-phenylpyridinium, TEA = tetraethylammonium.