Table 1.
Variability of Kt values for hOCT2 with transfection system (data from [35] and our laboratories).
| Compound | Kt (µM) |
Transfection system |
Reference |
|---|---|---|---|
| Dopamine | 1400 | cc | [53] |
| 390 | oo | [54] | |
| Histamine | 940 | cc | [53] |
| 1300 | oo | [54] | |
| MPP | 19 | oo | [55] |
| 7.8 | cc | [56] | |
| 12 | cc | Unpublished | |
| 3.1 | cc | [57] | |
| 12.3 | Unpublished | ||
| 19.5 | cc | [58] | |
| Norepinephrine | 1500 | cc | [53] |
| 1900 | oo | [54] | |
| Serotonin | 290 | cc | [53] |
| 80 | oo | [54] | |
| TEA | 27 | cc | [59] |
| 76 | oo | [55] | |
| 109 | cc | [60] | |
| 20 | cc | [61] | |
| 46 | cc | [17] | |
cc = cultured cell (HEK293 or CHO), oo = oocyte, MPP = 1-methyl-4-phenylpyridinium, TEA = tetraethylammonium.