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. 2012 Jan 21;3(3):252–256. doi: 10.1021/ml200304j

Table 1. Various Heterocyclic Substituted Diazepenes' Human Binding/Functional Activity and Mouse Functional BRS-3 Activity.

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a

Enantiomerically pure compounds unless otherwise noted.

b

Data expressed as mean ± SD (n ≥ 2 independent experiments).

c

%Act represents the maximum activation of tested compound relative to that of the known BRS-3 agonist dY peptide compound.