. 2012 May 30;3(7):574–578. doi: 10.1021/ml3000935

Table 1. Synthesis of Cyclic Sulfonimidamides 8c–f from Sulfinamide 6^a.

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Typical conditions: (1) 6, MeCN, N-chlorosuccinimide, 15 min at 0 °C, then amino acid reagent and DIPEA, rt; (2) sodium amylate, MeOH, reflux.

Isolated yields over two steps given in parentheses.

Table 1. Synthesis of Cyclic Sulfonimidamides 8c–f from Sulfinamide 6a.