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. Author manuscript; available in PMC: 2014 Nov 14.
Published in final edited form as: J Med Chem. 2013 Oct 28;56(21):8765–8780. doi: 10.1021/jm401232v

Table 1.

Single concentration screening of scaffolds 8 and 9 in the cytoprotection assay against HIV-1 in CEM-SS cells.

graphic file with name nihms532581u1.jpg
Compound R Inhibition % @ 10 μM Viability % @ 10 μM
8a graphic file with name nihms532581t1.jpg 7 85
9a 51 100
8b graphic file with name nihms532581t2.jpg 0 99
9b 17 90
8c graphic file with name nihms532581t3.jpg 5 100
9c 42 93
8d graphic file with name nihms532581t4.jpg 0 100
9d 88 95
8e graphic file with name nihms532581t5.jpg 0 100
9e 57 100
8f graphic file with name nihms532581t6.jpg 0 100
9f 10 99
8g H 5 100
9g 0 100