Table 5.
Compound | EC50 WT HIV (μM) | EC50 NNRTIr HIV (μM) | ratio NNRTIr/WT |
---|---|---|---|
9d | >5.0 | 2.4 | < 0.5 |
17d | 7.2 | 2.1 | 0.3 |
17f | 4.7 | 1.0 | 0.2 |
18a | 1.0 | 0.6 | 0.6 |
18e | 4.1 | 1.8 | 0.4 |
Compound | EC50 WT HIV (μM) | EC50 NNRTIr HIV (μM) | ratio NNRTIr/WT |
---|---|---|---|
9d | >5.0 | 2.4 | < 0.5 |
17d | 7.2 | 2.1 | 0.3 |
17f | 4.7 | 1.0 | 0.2 |
18a | 1.0 | 0.6 | 0.6 |
18e | 4.1 | 1.8 | 0.4 |