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. 2013 May 31;4(8):742–746. doi: 10.1021/ml400146c

Table 5. Pharmacokinetic Parameters for 2 in Rat and Dog.

species Cl (mL/min/kg) Vdss (L/kg) F (%)
rata,b 13 0.8 38
doga,c 1.1 0.2 89
a

Measured on the free base.

b

Average of 4 female rats; p.o. 5 mg/kg; i.v. 2 mg/kg.

c

Average of one male and one female; p.o. 2 mg/kg; i.v. 1 mg/kg.