Table 1. Antibacterial Activity of AA Series and Antibiotics on Enterobacterial Strains.
| MIC
(μM) |
||||
|---|---|---|---|---|
|
E. colia |
E. aerogenesb |
|||
| AG100 | AG100A | EA289 | EA298 | |
| molecules | WT | AcrAB-strain | MDR isolate | TolC-strain |
| Actc | >128 | 2 | >128 | 32 |
| Cipd | 0.125 | 0.03 | 64 | 8 |
| Flee | 0.5 | 0.125 | >128 | 16 |
| AA08 | 32 | 8 | 16 | 8 |
| AA23 | 16 | 8 | 16 | 8 |
| AA19 | 64 | 16 | >128 | 128–64 |
| AA24 | 64 | 64 | 128–64 | 64 |
| AA36 | 8 | 8 | 16 | 8 |
| AA37 | 16 | 8 | 8 | 4 |
| AA38 | 8 | 8 | 16 | 8 |
Laboratory strains.
Resistant clinical isolates.
Actinonin.
Ciprofloxacin.
Fleroxacin.