Table 1.
Log P values of radiolabeled NODAGA-E-[c(RGDfK)]2 determined by octanol/water partition assays
| Compound | Log Poctanol/PBS ± SD |
|---|---|
| Al18F-NODAGA-RGD2 | −4.26 ± 0.02 |
| 68Ga-NODAGA-RGD2 | −4.50 ± 0.01 |
| 111In-NODAGA-RGD2 | −4.34 ± 0.09 |
Log P values of radiolabeled NODAGA-E-[c(RGDfK)]2 determined by octanol/water partition assays
| Compound | Log Poctanol/PBS ± SD |
|---|---|
| Al18F-NODAGA-RGD2 | −4.26 ± 0.02 |
| 68Ga-NODAGA-RGD2 | −4.50 ± 0.01 |
| 111In-NODAGA-RGD2 | −4.34 ± 0.09 |