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. Author manuscript; available in PMC: 2014 May 29.
Published in final edited form as: Future Med Chem. 2011 Mar;3(3):367–390. doi: 10.4155/fmc.10.282

Table 1. Protein Data Bank codes, ligands and sources of crystal H structures of 11β-HSD1.

PDB code Ligand Source Ref.
Human 11β-HSD1
1XU7 9 Syrrx [35]
1XU9 9, 10 Syrrx [35]
2BEL 11 Biovitrum _
2ILT 12 Abbott [36]
2IRW 13 Abbott [37]
2RBE 17 Amgen & Biovitrum [38]
3BYZ 14 Amgen & Biovitrum [39]
3BZU 15 Amgen [40]
3CH6 18 Bristol-Myers Squibb [41]
3CZR 9, 20 Amgen [42]
3D3E 25 Amgen [43]
3D4N 21 Amgen [43,44]
3D5Q 19 Amgen [44]
3EY4 16 Amgen [45]
3FCO 26 Amgen [46]
3FRJ 24 Amgen [47]
3H6K 23 Wyeth [48]
3HFG 22 Wyeth [48]
Mouse 11β-HSD1
1Y5M - Amgen [49]
1Y5R 2b Amgen [49]
Guinea pig 11β-HSD1
1XSE - Biovitrum [50]
3DWF - University of Birmingham (UK) [51]
3G49 27 Pfizer [30]

No paper has been published describing the 2BEL structure.

11β-HSD1: 11β-hydroxysteroid dehydrogenase type 1; PDB: Protein Data Bank.