Table 1. Protein Data Bank codes, ligands and sources of crystal H structures of 11β-HSD1.
PDB code | Ligand | Source | Ref. |
---|---|---|---|
Human 11β-HSD1 | |||
1XU7 | 9 | Syrrx | [35] |
1XU9 | 9, 10 | Syrrx | [35] |
2BEL | 11 | Biovitrum | _† |
2ILT | 12 | Abbott | [36] |
2IRW | 13 | Abbott | [37] |
2RBE | 17 | Amgen & Biovitrum | [38] |
3BYZ | 14 | Amgen & Biovitrum | [39] |
3BZU | 15 | Amgen | [40] |
3CH6 | 18 | Bristol-Myers Squibb | [41] |
3CZR | 9, 20 | Amgen | [42] |
3D3E | 25 | Amgen | [43] |
3D4N | 21 | Amgen | [43,44] |
3D5Q | 19 | Amgen | [44] |
3EY4 | 16 | Amgen | [45] |
3FCO | 26 | Amgen | [46] |
3FRJ | 24 | Amgen | [47] |
3H6K | 23 | Wyeth | [48] |
3HFG | 22 | Wyeth | [48] |
Mouse 11β-HSD1 | |||
1Y5M | - | Amgen | [49] |
1Y5R | 2b | Amgen | [49] |
Guinea pig 11β-HSD1 | |||
1XSE | - | Biovitrum | [50] |
3DWF | - | University of Birmingham (UK) | [51] |
3G49 | 27 | Pfizer | [30] |
No paper has been published describing the 2BEL structure.
11β-HSD1: 11β-hydroxysteroid dehydrogenase type 1; PDB: Protein Data Bank.