Table 5.
IC50 values of 7-methoxyflavone derivatives from Kaempferia parviflora on PDE5 and PDE6 (n = 3).
Compound | IC50 (μM)
|
IC50 ratio PDE6/PDE5 | |
---|---|---|---|
PDE5 | PDE6 | ||
2 | 10.64 ± 2.09 | 39.45 ± 1.00 | 3.71 |
4 | 37.38 ± 1.15 | 27.33 ± 2.46 | 0.73 |
6 | 16.32 ± 1.93 | 42.58 ± 2.11 | 2.61 |
8 | 30.41 ± 2.34 | 7.83 ± 1.12 | 0.26 |
Dipyridamole | 1.46 ± 0.81 | 0.231 ± 0.03 | 0.16 |
Sildenafil | 0.0068 ± 0.00 | 0.033 ± 0.01 | 4.85 |