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. 2014 Mar 12;39(8):1843–1851. doi: 10.1038/npp.2014.31

Table 1. Binding Affinities for CSE and Nicotine at nAChRs.

nAChR subtype Region analyzed CSE Ki CSE 95% CI Nic Ki Nic 95% CI
α4β2 VPM/VPL thalamus 10.34 nM 7.7–13.8 nM 16.29 nM 11.2–23.8 nM
α3β4 Medial habenula 1.112 μM 0.75–1.66 μM 1.285 μM 0.85–1.86 μM
α3β2 Superior colliculus 0.0809 μM 0.024–0.272 μM 0.172 μM 0.032–0.921 μM
α7 Dentate gyrus 32.69 μM 19.6–54.5 μM 38.05 μM 21.42–67.62 μM