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. Author manuscript; available in PMC: 2014 Jun 23.
Published in final edited form as: J Med Chem. 2007 Mar 3;50(7):1442–1444. doi: 10.1021/jm061484y

Table 4.

Oral Pharmacokinetics of Compound 14 in the Rat at 10 mg/kg (0.75% Methocell/1% Tween).

Dose= 2 mg/kg
Tmax= 2.2 h
Cmax= 0.92 μg/mL
AUC= 6.10 μg• h/mL
t½= 4.2 h
CL= 0.52 L/h/kg
Vss= 0.6 L/kg
%F= 31