Table 3.
Drug | Lipophilicity | Distribution | Protein binding | Elimination |
---|---|---|---|---|
Cefazolin [30] | Low | Widely, to most tissues | 80% | Renal (60–80%) |
Tobramycin [30] | High | Mainly extracellular fluid | 0–30% | Renal (60–85%), mainly excretion, some secretion |
Gentamicin [31] | Intermediate | Mainly extracellular fluid | 0–30% | Renal (70–100%), mainly excretion, some secretion |
Vancomycin [32, 33] | Intermediate | Total body water and other tissues | 30–55% | Renal (40–100%) |