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. 2014 Jun 19;2014:848937. doi: 10.1155/2014/848937

Table 2.

Ki values of the BCPI mutants towards BCP.

Inhibitor Sequence Ki (nM)
Wild EQQSRLGLRLPAKKT 0.11 ± 0.006 [4]
Δ2 EQQSRLGLRLPAK 0.36 ± 0.037 [4]
Δ6 EQQSRLGLR 2.40 ± 0.19 [4]
Δ10 EQQSR nsi [4]
S75A EQQARLGLRLPAKKT
R76A EQQSALGLRLPAKKT
L77A/G78A EQQSRAALRLPAKKT 59.6 ± 10.7
L77A EQQSRAGLRLPAKKT 2.7 ± 1.54
G78A EQQSRLALRLPAKKT 5.58 ± 1.83
L79A/R80A EQQSRLGAALPAKKT 10.7 ± 6.82
L81A/P82A EQQSRLGLRAAAKKT

nsi: no significant inhibition.

∗Not significantly different from the wild.

[4]: Kurata et al., 2001.