Table 2.
Ki values of the BCPI mutants towards BCP.
| Inhibitor | Sequence | Ki (nM) |
|---|---|---|
| Wild | EQQSRLGLRLPAKKT | 0.11 ± 0.006 [4] |
| Δ2 | EQQSRLGLRLPAK | 0.36 ± 0.037 [4] |
| Δ6 | EQQSRLGLR | 2.40 ± 0.19 [4] |
| Δ10 | EQQSR | nsi [4] |
| S75A | EQQARLGLRLPAKKT | ∗ |
| R76A | EQQSALGLRLPAKKT | ∗ |
| L77A/G78A | EQQSRAALRLPAKKT | 59.6 ± 10.7 |
| L77A | EQQSRAGLRLPAKKT | 2.7 ± 1.54 |
| G78A | EQQSRLALRLPAKKT | 5.58 ± 1.83 |
| L79A/R80A | EQQSRLGAALPAKKT | 10.7 ± 6.82 |
| L81A/P82A | EQQSRLGLRAAAKKT | ∗ |
nsi: no significant inhibition.
∗Not significantly different from the wild.
[4]: Kurata et al., 2001.