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. 2014 May 13;5(7):760–765. doi: 10.1021/ml500053b

Table 4. Pharmacokinetic Parameters for 10i in Rat and Monkey.

species CL (mL/min/kg) Vdss (L/kg) F (%)
rata 47 14 81
monkeyb 27 16 39
a

Average of 3 male Sprague–Dawley rats; p.o. 10 mg/kg; i.v. 1 mg/kg.

b

Average of 3 male cynomolgus monkeys; p.o. 2 mg/kg; i.v. 0.5 mg/kg.