Table 2.
Activity of N,N-dimethylaminopropyl-substituted benzimidazoles 6 in the FRET assay.
Compound | R1 | EC50[μM]a |
---|---|---|
6h |
![]() |
160 ± 15 |
6i |
![]() |
160 ± 29 |
6j |
![]() |
290 ± 100 |
EC50 values are shown ± standard error from triplicate experiments.
Activity of N,N-dimethylaminopropyl-substituted benzimidazoles 6 in the FRET assay.
Compound | R1 | EC50[μM]a |
---|---|---|
6h |
![]() |
160 ± 15 |
6i |
![]() |
160 ± 29 |
6j |
![]() |
290 ± 100 |
EC50 values are shown ± standard error from triplicate experiments.