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. Author manuscript; available in PMC: 2015 May 26.
Published in final edited form as: Angew Chem Int Ed Engl. 2014 Apr 8;53(22):5600–5603. doi: 10.1002/anie.201310905

Table 3.

Tryptamine Scope.[a–e]

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[a]

Ar = 4–(t-Bu)C6H4.

[b]

Conditions: 4 (1 equiv), (R)–STRIP (10) (5 mol%), Na3PO4 (3 equiv), ArN2BF4 (1 equiv), MTBE, rt, 2–8 h.

[c]

Isolated yields.

[d]

ee determined by chiral phase HPLC.

[e]

Relative and absolute stereochemistry assigned by analogy to 5.