Table 2. Metabolic clearance of three compounds in rat and human.
Suspension are taken from Pfizer Research Technology Center values, LiverChip values are day 6 for rat (two experiments) and day 4 for human (four experiments).
Drug | Enzyme | Clearance values (µL per min, per million cells) |
|||
---|---|---|---|---|---|
Rat suspension | Rat LiverChip | Human suspension | Human LiverChip | ||
Midazolam | 3A4 | 35 | 38 | 13 | 13 |
Naloxone | Phase II | 51 | 39 | 30 | 29 |
Propranolol | 1A2, 2D6 | 61 | 48 | 19 | 8 |