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. 2014 Jun 23;13(14):2172–2191. doi: 10.4161/cc.29214

Table 3. Table of screened compounds which also inhibit the kinases that are more potently inhibited (>2-fold) by Bos-I compared with Dasatinib. (as identified in Table 2).

  Remaining Kinase activity (%)
  Bos-I Erlotinib Gefitinib Lapatinib Sunitinib
EGFR 3.84 4.21 2.97 8.02 89.17
HGK MAP4K4 1.03 76.48 97.78 111.21 12.44
MINK/MINK1 1.21 85.68 102.32 110.74 10.46
RET 18.94 48.57 76.94 99.77 3.43
ERBB4/HER4 1.53 61.41 24.15 11.19 94.81

Kinases inhibited by >50% are highlighted in red.