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. Author manuscript; available in PMC: 2014 Aug 14.
Published in final edited form as: Bioconjug Chem. 2012 Dec 4;23(12):2377–2385. doi: 10.1021/bc3003919

Table 1.

PSMA in Vitro Inhibitory Activitiesa

compound Ki (pM)
800CW-1 70 ± 5b
800CW-2 40 ± 10b
800CW-3 20 ± 5b
800RS-1 100 ± 10cd
800RS-2 200 ± 50b
800RS-3 4 ± 0.5c
ICG-1 700 ± 10cd
ICG-2 400 ± 60cd
ICG-3 200 ± 5cd
Cy7-1 1 ± 0.5c
Cy7-2 7 ± 0.4b
Cy7-3 5 ± 0.2c
Cy5.5-1 90 ± 40b
Cy5.5-2 50 ± 20b
Cy5.5-3 50 ± 2c
a

Values are in Ki ± SEM.

b

n = 4.

c

n = 2.

d

Measured in DMSO; all others in water.