Skip to main content
. Author manuscript; available in PMC: 2014 Aug 14.
Published in final edited form as: Biochem Pharmacol. 2013 Mar 13;85(10):1495–1503. doi: 10.1016/j.bcp.2013.02.039

Table 1.

The IC50 and h values of PPAR agonists and other TZDs.

Name IC50 (μM) h
PPARγ agonists AS-252424 4 2
Englitazone 7 1.6
A6335 8 1.2
Rosiglitazone 12 1.2
Cay10415 15 1.4
Darglitazone 25 1.4
AS605240 60 0.8
Pioglitazone 95 0.8
Troglitazone 100 0.8
Ciglitazone 120 0.7
PPARα agonists Fenofibrate 80 1.5
Gemfibrozil 290 0.9
PPARβ/δ agonists GW0742 80 1
GW501516 120 0.8
Other TZDs TZD +
CDS005865 >>100

Where h is the Hill coefficient.