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. Author manuscript; available in PMC: 2014 Aug 16.
Published in final edited form as: J Med Chem. 2010 Aug 12;53(15):5439–5448. doi: 10.1021/jm901808w

Table 3.

The growth inhibitory potency (IC50, uM) of GNF-7

TPR-Met-Ba/F3 NPM-ALK-Ba/F3 JAK1-Ba/F3 JAK2-Ba/F3 JAK2-V617F-Ba/F3 JAK3-Ba/F3 FGFR3-Ba/F3 Flt3-Ba/F3 Flt3-ITD-Ba/F3 PDGFRβ-Ba/F3 TrkC-Ba/F3 Colo205 SW620 U87 HEK293T
3.401 1.466 0.044 0.127 0.050 2.018 0.009 0.359 0.012 0.011 0.008 0.005 0.001 5.956 >10