Skip to main content
. 2014 Jul 8;57(15):6594–6609. doi: 10.1021/jm5006176

Table 4. Selectivity of 11a-1 against a Panel of PTPs.

graphic file with name jm-2014-006176_0011.jpg

PTP IC50 (μM) PTP IC50 (μM)
SHP2 0.20 ± 0.02 VHR 3.2 ± 0.1
LYP 1.05 ± 0.02 PTPμ 3.3 ± 0.2
HePTP 1.03 ± 0.08 STEP 4.0 ± 0.2
PTPH1 1.07 ± 0.07 PEZ 5.3 ± 0.2
SHP1 1.44 ± 0.04 PTPσ 8.6 ± 0.4
Ssu72 1.3 ± 0.2 UBLCP1 9.7 ± 0.5
PTP1B 2.29 ± 0.03 laforin 12.2 ± 2
LMWPTP 2.34 ± 0.02 CDC14A 16 ± 4
VHZ 2.3 ± 0.2 PTPε >20
PTPγ 2.4 ± 0.4 PTPα >100
MKP5 2.9 ± 0.1