Table 1.
| Agent | Target (IC50) |
|---|---|
| AMG900 | Aurora A (5 nM) |
| Aurora B (4 nM) | |
| Aurora C (1nM) | |
| MLN8237 | Aurora A (61 nM) |
| AZD1152 | Aurora A (1369 nM) |
| Aurora B (.36 nM) | |
| Aurora C (17 nM) | |
| PHA-739358 | Aurora A (13 nM) |
| Aurora B (79 nM0 | |
| Aurora C (61 nM) | |
| Tozasertib | Aurora A (0.6 nM) |
| Aurora B (18 nM) | |
| Aurora C (4.5 nM) | |
| AT9283 | Aurora A (3 nM) |
| Aurora B (3 nM) | |
| ENMD2076 | Aurora A (13 nM) |
| Aurora B (350 nM) |