Table 2.
Activity of aza-analogues with C-1 homologues as standards [IC50 (μM)]
Cell line |
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---|---|---|---|---|---|
HeLa (cervical cancer) | <0.4 μM | <0.4 μM | Non-inhibitory | >100 μM | >100 μM |
MCF7 (breast cancer) | <0.4 μM | <0.4 μM | Non-inhibitory | >100 μM | >100 μM |