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. Author manuscript; available in PMC: 2014 Sep 5.
Published in final edited form as: Chem Rev. 2013 Jun 17;113(8):5701–5765. doi: 10.1021/cr4000144

Table 3.

Synthesis of Tricyclic Bridged Lactams via Domino Diels-Alder/Schmidt Reaction by Aubé

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entry ketoazide 175 R1 R2 yield of
176 (%)		 yield of
177 (%)
1 175a (CH2)2OBn H 43 24
2 175b 4-Br-C6H4 H 43 23
3 175c C6H5 H 46 23
4 175d H H 41 22
5 175e H i-Pr 43 28
6 175f H Ph 85 0