Table 2.
Reaction Scope with Respect to Arylamides [a]
![]() | |||
---|---|---|---|
Entry | Ar | Product | Yield, % |
1 | C6H5 | ![]() |
78 |
2 | 4-CF3C6H4 | ![]() |
70 |
3 | 4-BrCC6H4 | ![]() |
73 |
4 | 4-NO2C6H4 | ![]() |
78 |
5 | 2-MeC6H4 | ![]() |
86 |
6 | 3-IC6H4 | ![]() |
84 |
7[b] | 2-MeOC6H4 | ![]() |
74 |
8[c] | 2-furyl | ![]() |
81 |
9[d] | 2-thiophenyl | ![]() |
86 |
Amide 0.5 mmol, CF3CH2OH 5 mL, air. Yields are isolated yields. Please see Supporting information for details.
Time: 18 h.
Time: 16 h.
Time: 20 h.