Table 3.
Scope of Propargylic Alcohols 9a
| Entry | Substrate
|
Product
|
Yield (%)b |
|---|---|---|---|
| 1 | 11a, R = nBu | 12a | 72 |
| 2 | 11b, R = iPr | 12b | 83 |
| 3 | 11c, R = Ph | 12c | 42 |
| 4 |
![]() 11d |
![]() 12d |
60 |
| 5 |
![]() 11e |
![]() 13 |
63c |
Conditions: 9 (1 equiv), indole 8a (2 equiv), Cu(CH3CN)4PF6 (10 mol %), 60 °C, ClCH2CH2Cl.
Isolated yield.
Indole 8b was employed.



