Table 1. Kinetic parameters of the binding of luteolin to VRK1.
Ka(M−1S−1) | Kd(S−1) | KD | |
Luteolin | 43.62 | 0.0464 | 5.8 µM |
Eupatiln | 414 | 0.0763 | 184 µM |
Wogonin | 51.72 | 0.083 | 120 µM |
Ka(M−1S−1) | Kd(S−1) | KD | |
Luteolin | 43.62 | 0.0464 | 5.8 µM |
Eupatiln | 414 | 0.0763 | 184 µM |
Wogonin | 51.72 | 0.083 | 120 µM |