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. 2014 Aug 26;11(9):8709–8742. doi: 10.3390/ijerph110908709

Table 4.

ERβ selective compounds with their respective fold selectivity for ERβ. * Data for assays performed: the first number indicates data for ERβ and the second number indicates data for ERα; In superscript, B indicates binding assays, R indicates HEK 293 reporter gene assays. NA indicates where binding data is not available but functional data discussed in main text. ID indicates the compound number that is cited in the text.

ID Structure Ref Fold Selectivity Data *
10 graphic file with name ijerph-11-08709-i010.jpg [80] 2.2 B
68.4 R
(RBA: 107/48) B
(>5400 nM/79 nM) R
11 graphic file with name ijerph-11-08709-i011.jpg [125] 0.54 B (RBA: 0.038/0.07) B
12 graphic file with name ijerph-11-08709-i012.jpg [125] 1.56 B (RBA:0.056/0.036) B
13 graphic file with name ijerph-11-08709-i013.jpg [124] NA NA
14 graphic file with name ijerph-11-08709-i014.jpg [126] 8.2 B (RBA: 61.1/7.8) B
15 graphic file with name ijerph-11-08709-i015.jpg [126] 10.1 B (RBA: 49.9/4.9) B
16 graphic file with name ijerph-11-08709-i016.jpg [127] 7.4 B (87/11.8) B