Skip to main content
. Author manuscript; available in PMC: 2014 Oct 27.
Published in final edited form as: J Am Chem Soc. 2013 Mar 11;135(11):4333–4363. doi: 10.1021/ja3109664

Scheme 7.

Scheme 7

Sulfonylation reactions on solid phase. Sulfonates were subsequently modified on solid phase (Scheme 8) or were subjected to TFA cleavage/deprotection and purified and analyzed in aqueous solution.a

a RN′ = Ac-Thr(OtBu)-Tyr(OtBu)-, RC′ = -Asn(Trt)-NHRink-Resin. RN = Ac-Thr-Tyr-, RC = -Asn-NH2.