Targets | Ligands | |
---|---|---|
5-HT1A receptor | 5-HT | Olanzapine |
5-HT1B receptor | Dopamine | Pimozide |
5-HT2A receptor | Noradrenaline | Quetiapine |
5-HT2C receptor | Amphetamine | Reboxetine |
5-HT3 receptor | α-MSH | Risperidone |
5-HT4 receptor | Aripiprazole | Sertraline |
5-HT6 receptor | Bupropion | Sibutramine |
α1 adrenoceptor | meta-Chlorophenylpiperazine | Sulpiride |
α2 adrenoceptor | Chlorpromazine | Δ9-tetrahydrocannabinol, THC |
β2 adrenoceptor | Cyproheptadine | Topiramate |
CRF1 receptor | DAMGO | |
Dopamine D1 receptor | Desipramine | |
Dopamine D2 receptor | Fenfluramine | |
Dopamine D3 receptor | Fluoxetine | |
Dopamine D4 receptor | cis-Flupenthixol | |
Ghrelin receptor (GHS-R1a) | Fluvoxamine | |
μ opioid receptor | Ghrelin | |
Melanocortin MC1 receptor | Haloperidol | |
NET, noradrenaline transporter | Leptin | |
SERT, 5-HT transporter | Neuropeptide Y |
This Table lists the protein targets and ligands in this article which are hyperlinked to corresponding entries in http://www.guidetopharmacology.org, the common portal for data from the IUPHAR/BPS Guide to PHARMACOLOGY (Pawson et al., 2014) and the Concise Guide to PHARMACOLOGY 2013/14 (Alexander et al., 2013a–c).