Table 2.
Ligand | Kinetic parameters | Ref. | |
---|---|---|---|
(A) | Stearic acid | ND | [28] |
Palmitic acid | ND | [28] | |
Cholesterol | ND | [28] | |
Lauric acid | ND | [28] | |
Triacylglycerols | ND | [28] | |
Fatty alcohols | ND | [28] | |
(B) | Retinol | Kd ~ 0.6 μM | [8] |
Oleic acid | ND | [46] | |
16-APa | Kd ~ 0.8 μM | [29] | |
DAUDAb | Ki ~ 2.8 μM | [29] | |
Cholesterol | Ki ~ 15.9 μM | [29] | |
Lauric acid | Ki ~ 9.1 μM | [29] | |
Palmitic acid | Ki ~ 3.2 μM | [29] | |
Stearic acid | Ki ~ 1.3 μM | [29] | |
Phosphatidylcholine | Ki ~ 1.2 μM | [29] |
16-AP, 16-(9-anthroyloxy)palmitic acid.
DAUDA, 11-(5-dimethylamino-1-naphthalenylsulphonyl)amino-undecanoic acid.