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. 2014 May 13;9(7):1536–1544. doi: 10.1021/cb5001586

Table 1. SAR Analysis of Eastern Analogues.

graphic file with name cb-2014-001586_0006.jpg

analog R μM
3 4-Cl 0.04 ± 0.01
7 H 0.30 ± 0.02
8 2-OCH3 0.40 ± 0.08
9 4-F 0.07 ± 0.02
10 4-CF3 0.39 ± 0.10
11 2-OCH3 1.7 ± 0.6
12 2-Cl, 4-Cl 0.25 ± 0.04
13 2-F, 4-Cl 0.06 ± 0.02
a

Average of at least three replicates ± standard deviation.