Figure 2.
In vitro binding and inhibition studies. (A) IC50 value of Cu-E4-Fl 6, measured via a competitive binding assay using HEK-hGLP1R cells. (B) Confocal microscopy imaging experiments using 916–1 insulinoma cells.
In vitro binding and inhibition studies. (A) IC50 value of Cu-E4-Fl 6, measured via a competitive binding assay using HEK-hGLP1R cells. (B) Confocal microscopy imaging experiments using 916–1 insulinoma cells.