Table 2. Antagonism of NT Induced Calcium Release at NTS1 Compared to Target Compound Induced Calcium Mobilization and Binding Affinity at NTS2 for 7-Chloroquinolyl (A), Naphthyl (B), and 4-F-Phenyl (C) Substituted Pyrazole Carboxamides at the NTS1 and NTS2 Receptors.

^a[¹²⁵I]NT.

^bEC₅₀, K_e, IC₅₀, and K_i values are all nM ± SEM.

^cE_max value is % 5b.

^dNot active.