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. 2014 Jun 11;136(28):10139–10147. doi: 10.1021/ja5049303

Table 3. Tandem C–H Fluorination and SNAra.

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a

Isolated yields from the two-step sequence for reactions performed with 0.2 mmol of heteroarene. Yields in parentheses were determined by 19F NMR spectroscopy for the independent fluorination reaction.

b

The isolated product contained ∼5% of an inseparable impurity.

c

The Boc group was cleaved during the SNAr reaction.