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. 2014 Nov 12;9(11):e110502. doi: 10.1371/journal.pone.0110502

Table 1. Half-maximal effective concentration (EC50) for selected ligands at NK1R or CCK2R.

NK1R CCK2R
Ligand EC50 (nM) Ligand EC50 (nM)
s-SubP-NH2 1.4 s-CCK4-NH2 4.9
l-SubP-NH2 0.4 l-CCK4-NH2 2.6
s-SubP-COOH 449.3 s-CCK4-Gly-COOH >1000
l-SubP-COOH 6.1 l-CCK4-Gly-COOH >1000

All values represent the mean from at least three independent experiments, each performed in triplicate.