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. Author manuscript; available in PMC: 2014 Nov 14.
Published in final edited form as: Clin Cancer Res. 2009 Mar 17;15(7):2380–2386. doi: 10.1158/1078-0432.CCR-08-2387

Table 1.

Structure and inhibition constants (Ki) for CXCR1 and CXCR2

graphic file with name nihms-352988-t0001.jpg
KiCXCR2 (nmol/L) KiCXCR1 (nmol/L) Ratio
SCH-527123 0.05 3.7 74
SCH-479833 0.17 7 100