. 2014 Aug 22;57(21):8860–8879. doi: 10.1021/jm500942v

Table 1. 3-Alkylphenyl-4(1H)-quinolones^a.

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Dihydroartemisinin (DHA), chloroquine (CQ), and atovaquone (ATO) are internal controls for each in vitro assay: DHA, 5.5 nM W2 and 5.9 nM TM90-C2B; CQ, 229 nM for TM90-C2B and 421 nM for W2; and ATO, 1.4 nM W2 and 18.4 μM TM90-C2B.

Table 1. 3-Alkylphenyl-4(1H)-quinolonesa.

Table 1. 3-Alkylphenyl-4(1H)-quinolones^a.