Table 1.
Specificity of biochanin A against mitogen-activated kinase related kinases.
Kinase | Relative kinase activity (% of untreated control) |
---|---|
ASK1 (h) | 103 ± 0 |
c-RAF (h) | 86 ± 10 |
JNK1α1 (h) | 98 ± 2 |
MAPK1 (h) | 89 ± 4 |
MEK1 (h) | 75 ± 7 |
MKK4 (m) | 104 ± 3 |
MKK6 (h) | 109 ± 5 |
MKK7β (h) | 89 ± 6 |
MSK1 (h) | 85 ± 5 |
PKBα (h) | 101 ± 8 |
Rsk2 (h) | 80 ± 5 |
SAPK2a (h) | 88 ± 3 |
TAK1 (h) | 91 ± 6 |
TAO1 (h) | 80 ± 1 |
TAO2 (h) | 84 ± 5 |